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PJ34

●Purchase●DescriptionAcell-permeable,water-soluble,potentinhibitorofpoly(ADP-ribose)polymerase(PARP;EC50=20nM)

产品型号:27041

更新时间:2024-11-25

  • 详细介绍
  • 品牌BPS Bioscience
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Description

A cell-permeable, water-soluble, potent inhibitor of poly(ADP-ribose) polymerase (PARP; EC50 = 20 nM). Shown to be about 10,000 times more potent than the prototypical PARP inhibitor, 3-Aminobenzamide (Cat. No. 165350; EC50 = 200 µM). Does not act as an antioxidant at higher concentrations (1 µM to 10 mM). Exhibits neuroprotection in in vivo and in vitro models of stroke.

Synonyms
N-(5,6-Dihydro-6-oxo-2-phenanthridi­nyl)-2-acetamide hydrochloride

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