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PYR-41

●Purchase●DescriptionPYR-41isacellpermeable

产品型号:27716-1

更新时间:2024-11-28

  • 详细介绍
  • 品牌BPS Bioscience
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Description

PYR-41 is a cell permeable, irreversible inhibitor of ubiquitin activating enzyme E1 with little or no activity against E2s or E3s (IC50 < 10 μM). It blocks degradation of p53 and inhibits NF-kappaB-dependent pathways. PYR-41 also increases SUMOylation of proteins.

Synonyms
4–[4–[(5–Nitro–2–furanyl)methylene]?–3,5–dioxo–1–pyrazolidinyl]benzoic acid ethyl ester

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