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K252a

●Purchase●DescriptionK252aisageneralkinaseinhibitorthatinhibitsPKA(Ki=18nM),PKC(Ki=25nM),PKG(Ki=20nM),CaMK(Ki=1

产品型号:27033

更新时间:2024-11-29

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Description

K252a is a general kinase inhibitor that inhibits PKA (Ki = 18 nM), PKC (Ki = 25 nM), PKG (Ki = 20 nM), CaMK (Ki = 1.8 nM), and phosphorylase kinase (IC50 = 1.7 nM). It functions by acting competitively with ATP and noncompetitively with the substrate.

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