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Fasudil

●Purchase●DescriptionMonohydrochlorideformofHA-1077

产品型号:27029

更新时间:2024-11-29

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Description

Monohydrochloride form of HA-1077. Inhibits a number of kinases, including ROCK I (IC50 = 10.7 µM), ROCK II (IC50 = 1.9 µM), MAPK1 (IC50 = 5 µM), and PKCRK2 (IC50 = 4 µM). Weaker inhibitor of PKC (IC50 = 425 µM) and MLCK (IC50 = 95 µM) .

This product has been cited 2 times.

Synonyms
HA-1077, Monohydrochloride Salt, 1-(5-Isoquinolinesulfonyl)homopiperazine, HCl, Eril, AT-877

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