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CHIR-99021 (CT99021)

●Purchase●DescriptionCHIR-99021isahighlyspecificglycogensynthasekinase-3(GSK-3)inhibitorthatcaninhibitbothisoformswithIC50of10nM(GSK-3)and6

产品型号:27614-3

更新时间:2024-11-29

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Description

CHIR-99021 is a highly specific glycogen synthase kinase-3 (GSK-3) inhibitor that can inhibit both isoforms with IC50 of 10 nM (GSK-3α) and 6.7 nM (GSK-3β).

This product has been cited 1 time.

Synonyms
CHIR-99021; CT99021; 6-[2-[[4-(2,4-dichlorophenyl)-5-(5-methyl-1H-imidazol-2-yl)pyrimidin-2-yl]amino]ethylamino]pyridine-3-carbonitrile

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