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UNC0321 (TFA salt)

●Purchase●DescriptionUNC0321(trifluoroacetatesalt)isaselectivehistonelysinemethyltransferase(HMTase)inhibitorforG9aandGLP(alsoknownasEHMT1),withIC50of6nMand15nM,respectively

产品型号:27306

更新时间:2024-11-25

  • 详细介绍
  • 品牌BPS Bioscience
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Description

UNC0321 (trifluoroacetate salt) is a selective histone lysine methyltransferase (HMTase) inhibitor for G9a and GLP (also known as EHMT1), with IC50 of 6 nM and 15 nM, respectively. It is more than 40,000-fold more selective for G9a and GLP vs. SET7/9, SET8, PRMT3, or JMJD2E.

Synonyms
4-Quinazolinamine, 7-[2-[2-(dimethylamino)ethoxy]ethoxy]-2-(hexahydro-4-methyl-1H-1,4-diazepin-1-yl)-6-methoxy-N-(1-methyl-4-piperidinyl)-, trifluoroacetate

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